PDB
Resolution
2.8 Å
Released
July 8, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
BMS-986187
Ago-PAM
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
BMS-986187 L97 2.52x52 TM2 hydrophobic
BMS-986187 L119 3.23x23 TM3 Van der Waals
BMS-986187 A123 3.27x27 TM3 hydrophobic
BMS-986187 S126 3.30x30 TM3 Van der Waals
BMS-986187 I127 3.31x31 TM3 hydrophobic
BMS-986187 Y130 3.34x34 TM3 hydrophobic
BMS-986187 N131 3.35x35 TM3 polar (hydrogen bond)
BMS-986187 S177 4.54x54 TM4 Van der Waals
BMS-986187 G180 4.57x57 TM4 Van der Waals
BMS-986187 V181 4.58x58 TM4 hydrophobic
BMS-986187 M184 4.61x61 TM4 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 V T R P R D G A V V C M L Q F P S ECL2ICL3 R L L S G ICL3ECL3 D I D R R ECL3N-term M E P A P S A G A E L Q P P L F A N A S D A Y P S A C P S A G A N A S G P P N-termC-term P C G R P D P S S F S R A R E A T A R E R V T A C T P S D G P G G G A A A C-term G A R S A S S L A L A I A I T A L Y S A V C A V G L L G N V L V M F G I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S A K Y L M E G E L L C K A V L S I D Y Y N M F T S I F T L T M M S V D R Y I A V C H T P A K A K L I N I C I W V L A S G V G V P I M V M A P S W Y W D T V T K I C V F L F A F V V P I L I I T V C Y G L M L L R L R S V S K E K D R S L R R I T R M V L V V V G A F V V C W A P I H I F V I V W T L V D P L V V A A L H L C I A L G Y A N S S L N P V L Y A F L D E N F R Q F K R C L C R K
Helix box plot — Download: PNG | SVG V N G L L G V A C V A S Y L A T I A I A 1 F N L A L A D A L A T S T L P F Q S A K 2 M T L T F I S T F M N Y Y D I S L V A K 3 A K L I N I C I W V L A S G V G V P I M 4 Y C V T I I L I P V V F A F L F V C I K T 5 L V V V G A F V V C W A P I H I F V I V 6 V P N L S S N A Y G L A I C L H L A A 7

GPCRdb(A)
GPCRdb(A)
δ receptor
TM2
2x52 2.52x52 L97
TM3
3x23 3.23x23 L119
3x27 3.27x27 A123
3x30 3.30x30 S126
3x31 3.31x31 I127
3x34 3.34x34 Y130
3x35 3.35x35 N131
TM4
4x54 4.54x54 S177
4x57 4.57x57 G180
4x58 4.58x58 V181
4x61 4.61x61 M184