vapreotide
SMILES | None |
InChIKey | SWXOGPJRIDTIRL-UHFFFAOYSA-N |
Sequence | FCYWKVCW |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Surrogate |
Approved drug | Yes |
Database connections
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
SST2 | SSR2 | Human | Somatostatin | A | pKi | 8.3 | 9.2 | 10.1 | Guide to Pharmacology |
SST5 | SSR5 | Human | Somatostatin | A | pKi | 7.3 | 8.25 | 9.2 | Guide to Pharmacology |
SST5 | SSR5 | Rat | Somatostatin | A | pKi | 8.2 | 8.2 | 8.2 | Guide to Pharmacology |
SST2 | SSR2 | Rat | Somatostatin | A | pKi | 9.1 | 9.1 | 9.1 | Guide to Pharmacology |
SST3 | SSR3 | Rat | Somatostatin | A | pKi | 7.1 | 7.1 | 7.1 | Guide to Pharmacology |
SST2 | SSR2 | Mouse | Somatostatin | A | pKi | 6.1 | 7.65 | 9.2 | Guide to Pharmacology |
SST1 | SSR1 | Human | Somatostatin | A | pKi | 6.0 | 6.68 | 7.08 | PDSP Ki database |
SST2 | SSR2 | Human | Somatostatin | A | pKi | 8.27 | 9.43 | 10.3 | PDSP Ki database |
SST3 | SSR3 | Human | Somatostatin | A | pKi | 7.37 | 7.64 | 7.91 | PDSP Ki database |
SST4 | SSR4 | Human | Somatostatin | A | pKi | 6.45 | 6.93 | 7.35 | PDSP Ki database |
SST5 | SSR5 | Human | Somatostatin | A | pKi | 7.27 | 8.36 | 9.15 | PDSP Ki database |
SST5 | SSR5 | Rat | Somatostatin | A | pKi | 8.17 | 8.48 | 8.8 | PDSP Ki database |
SST3 | SSR3 | Mouse | Somatostatin | A | pKi | 7.64 | 7.64 | 7.64 | PDSP Ki database |
SST4 | SSR4 | Mouse | Somatostatin | A | pKi | 6.77 | 6.77 | 6.77 | PDSP Ki database |
SST2 | SSR2 | Mouse | Somatostatin | A | pKi | 6.1 | 8.45 | 10.0 | PDSP Ki database |
SST2 | SSR2 | Rat | Somatostatin | A | pKi | 9.07 | 9.07 | 9.07 | PDSP Ki database |
SST3 | SSR3 | Rat | Somatostatin | A | pKi | 7.06 | 7.06 | 7.06 | PDSP Ki database |
SST1 | SSR1 | Human | Somatostatin | A | pKi | 6.8 | 6.8 | 6.8 | ChEMBL |
SST2 | SSR2 | Human | Somatostatin | A | pKi | 10.1 | 10.1 | 10.1 | ChEMBL |
SST3 | SSR3 | Human | Somatostatin | A | pKi | 7.7 | 7.7 | 7.7 | ChEMBL |
SST3 | SSR3 | Human | Somatostatin | A | pKi | 7.4 | 7.65 | 7.9 | Guide to Pharmacology |
SST4 | SSR4 | Human | Somatostatin | A | pKi | 6.8 | 6.8 | 6.8 | ChEMBL |
SST5 | SSR5 | Human | Somatostatin | A | pKi | 8.3 | 8.3 | 8.3 | ChEMBL |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |