Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
AssayType |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
| 3404 | 6801 | 29 | None | 107 | 3 | Mouse | 9.6 | pEC50 | = | 9.6 | Functional | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | ||
| 5283155 | 6801 | 29 | None | 107 | 3 | Mouse | 9.6 | pEC50 | = | 9.6 | Functional | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | ||
| 5508 | 6801 | 29 | None | 107 | 3 | Mouse | 9.6 | pEC50 | = | 9.6 | Functional | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | ||
| CHEMBL1526258 | 6801 | 29 | None | 107 | 3 | Mouse | 9.6 | pEC50 | = | 9.6 | Functional | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | ||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Similar- ity |
Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
Assay Type |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
| 3404 | 6801 | 29 | None | - | 1 | Mouse | 8.3 | pKd | = | 8.3 | Binding | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5283155 | 6801 | 29 | None | - | 1 | Mouse | 8.3 | pKd | = | 8.3 | Binding | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5508 | 6801 | 29 | None | - | 1 | Mouse | 8.3 | pKd | = | 8.3 | Binding | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| CHEMBL1526258 | 6801 | 29 | None | - | 1 | Mouse | 8.3 | pKd | = | 8.3 | Binding | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||