Ligand source activities (1 row/activity)



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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Potency)		 # tested GPCRs
(Potency)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI
131648253 2991 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 2991 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 2991 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
131648253 2991 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 2991 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 2991 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
32051 4087 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960
566 4087 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960


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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Affinity)		 # tested GPCRs
(Affinity)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI
9140 2990 0 None - 1 Mouse 8.1 pKd = 8.1 Binding
N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.
Guide to Pharmacology None None None None 27117253