PDB
Resolution
3.2 Å
Released
Nov. 19, 2025
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
Chemerin
Agonist

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Ligand Amino Acid Generic Number Segment Interaction Type
Chemerin F86 2.53x53 TM2 Van der Waals
Chemerin Y93 2.60x60 TM2 hydrophobic
Chemerin Y93 2.60x60 TM2 aromatic (edge-to-face)
Chemerin Y96 2.63x63 TM2 Van der Waals
Chemerin F101 ECL1 hydrophobic
Chemerin F101 ECL1 aromatic (edge-to-face)
Chemerin S114 3.29x29 TM3 polar (hydrogen bond)
Chemerin A117 3.32x32 TM3 Van der Waals
Chemerin Q118 3.33x33 TM3 Van der Waals
Chemerin A172 4.60x60 TM4 Van der Waals
Chemerin R176 ECL2 polar (charge-charge)
Chemerin V179 ECL2 hydrophobic
Chemerin F181 ECL2 hydrophobic
Chemerin L186 ECL2 hydrophobic
Chemerin Y188 45.51x51 ECL2 hydrophobic
Chemerin N189 45.52x52 ECL2 hydrophobic
Chemerin N189 45.52x52 ECL2 polar (hydrogen bond)
Chemerin Q192 ECL2 polar (hydrogen bond)
Chemerin H203 5.35x36 TM5 Van der Waals
Chemerin Y262 6.51x51 TM6 hydrophobic
Chemerin Y262 6.51x51 TM6 aromatic (edge-to-face)
Chemerin H273 6.62x62 TM6 Van der Waals
Chemerin S278 ECL3 Van der Waals
Chemerin H280 ECL3 Van der Waals
Chemerin I286 7.35x34 TM7 hydrophobic
Chemerin T290 7.39x38 TM7 hydrophobic
Chemerin F294 7.43x42 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 K K ICL1ECL1 F H W P F ECL1ICL2 P V L S H R H R ICL2ECL2 D T V E F N N H T L C Y N N F Q K H D P D ECL2ICL3 I L I ICL3ECL3 H N S Y S ECL3N-term M E D L E E T L F E E F E N Y S Y D L D Y Y S L E S D L E E K V Q L N-termC-term A E I L K Y T L W E V S C S G T V S E Q L R N S E T K N L C L L E T A Q C-term G V V H W V S L V L Y C L A F V L G I P G N A I V I W F T G F K W T V T T L W F L N L A I A D F I F L L F L P L Y I S Y V A M N G I W L C K A N S F T A Q L N M F A S V F F L T V I S L D H Y I H L I H T L K N S L I V I I F I W L L A S L I G G P A L Y F R L T L I R H H V L T W V K F I I G Y L F P L L T M S I C Y L C L I F K V K K R S S S R H F W T I L V V V V A F V V C W T P Y H L F S I W E L T I H H H V M Q A G I P L S T G L A F L N S C L N P I L Y V L I S K K F R S F Q A R S V
Helix box plot — Download: PNG | SVG A N G P I G L V F A L C Y L V L S V W H 1 L N L A I A D F I F L L F L P L Y I S Y 2 V T L F F V S A F M N L Q A T F S N A K 3 S L I V I I F I W L L A S L I G G P A L 4 Y C I S M T L L P F L Y G I I F K V W T L 5 L V V V V A F V V C W T P Y H L F S I W 6 I P N L C S N L F A L G T S L P I G A 7

GPCRdb(A)
GPCRdb(A)
chemerin receptor 2
TM2
2x53 2.53x53 F86
2x60 2.60x60 Y93
2x63 2.63x63 Y96
TM3
3x29 3.29x29 S114
3x32 3.32x32 A117
3x33 3.33x33 Q118
TM4
4x60 4.60x60 A172
ECL2
45x51 45.51x51 Y188
45x52 45.52x52 N189
TM5
5x36 5.35x36 H203
TM6
6x51 6.51x51 Y262
6x62 6.62x62 H273
TM7
7x34 7.35x34 I286
7x38 7.39x38 T290
7x42 7.43x42 F294