GPCR CLASS (FAMILY)
Class A (Rhodopsin)
GPCR SPECIES
Homo sapiens
GPCR PREFERRED CHAIN
F
G PROTEIN (FAMILY)
Gi/o
G PROTEIN SPECIES
Homo sapiens
PDB CODE
RESOLUTION
3.5 Å
PUBLICATION DATE
May 27, 2026
LIGAND INTERACTIONS
LIGANDS
DAMGO - Agonist pubchem gtoplig chembl_ligand pubchem ,
BMS-986187 - PAM pubchem gtoplig chembl_ligand
PHYSIOLOGICAL LIGANDS
[Met]enkephalin (Human), dynorphin A-(1-8) (Human), dynorphin A (Human), dynorphin A-(1-13) (Human), β-endorphin (Mouse), endomorphin-1 (Human), β-endorphin (Rat), dynorphin B (Human), β-endorphin (Human), [Leu]enkephalin (Human), endomorphin-2 (Human)