Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
gasr_human 6.51x51 349 TM6 V => L N/A N/A Kopin AS et al (1994)
gasr_human 7.33x32 370 TM7 A => I N/A N/A Kopin AS et al (1995)
gasr_human 1.58x58 80 TM1 G => I N/A N/A Kopin AS et al (1995)
gasr_human 1.34x34 56 TM1 I => V N/A N/A Kopin AS et al (1995)
gasr_human 1.51x51 73 TM1 M => T N/A N/A Kopin AS et al (1995)
gasr_human 1.37x37 59 TM1 T => L N/A N/A Kopin AS et al (1995)
gasr_human 1.41x41 63 TM1 V => L N/A N/A Kopin AS et al (1995)
gasr_human 2.41x41 91 TM2 A => I N/A N/A Kopin AS et al (1995)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 3.47x47 149 TM3 A => S N/A N/A Kopin AS et al (1995)
gasr_human 3.27x27 129 TM3 A => T N/A N/A Kopin AS et al (1995)
gasr_human 3.31x31 133 TM3 L => F N/A N/A Kopin AS et al (1995)
gasr_human 3.29x29 131 TM3 S => T N/A N/A Kopin AS et al (1995)
gasr_human 3.28x28 130 TM3 V => T N/A N/A Kopin AS et al (1995)
gasr_human 3.34x34 136 TM3 V => T N/A N/A Kopin AS et al (1995)
gasr_human 4.51x51 180 TM4 L => C N/A N/A Kopin AS et al (1995)
gasr_human 4.47x47 176 TM4 V => A N/A N/A Kopin AS et al (1995)
gasr_human 5.55x55 235 TM5 A => M N/A N/A Kopin AS et al (1995)
gasr_human 5.49x49 229 TM5 I => T N/A N/A Kopin AS et al (1995)
gasr_human 5.45x46 225 TM5 L => I N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => Q N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => H N/A N/A Kopin AS et al (1995)
gasr_human 6.49x49 347 TM6 L => M N/A N/A Kopin AS et al (1995)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 6.52x52 350 TM6 Y => F N/A N/A Kopin AS et al (1995)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Beinborn M et al (1993)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Kopin AS et al (1995)
gasr_human 6.51x51 349 TM6 V => L N/A N/A Beinborn M et al (1993)
gasr_human 7.46x46 383 TM7 A => S N/A N/A Kopin AS et al (1995)
gasr_human 7.44x43 381 TM7 A => T N/A N/A Kopin AS et al (1995)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Kopin AS et al (1994)
gasr_human 1.60x60 82 TM1 S => D N/A N/A Wu SV et al (1999)
gasr_human 1.60x60 82 TM1 S => T N/A N/A Wu SV et al (1999)
gasr_human 1.60x60 82 TM1 S => A N/A N/A Wu SV et al (1999)
gasr_human 1.39x39 61 TM1 Y => A N/A N/A Blaker M et al (2000)
gasr_human 2.60x59 110 TM2 F => A N/A N/A Blaker M et al (2000)
gasr_human 2.61x60 111 TM2 T => A N/A N/A Blaker M et al (2000)
gasr_human 3.29x29 131 TM3 S => A N/A N/A Blaker M et al (2000)
gasr_human 3.33x33 135 TM3 G => A N/A N/A Blaker M et al (2000)
gasr_human 4.57x57 186 TM4 M => A N/A N/A Blaker M et al (2000)
gasr_human 4.64x65 193 TM4 T => A N/A N/A Blaker M et al (2000)
gasr_human 5.39x40 219 TM5 S => A N/A N/A Blaker M et al (2000)
gasr_human 5.46x461 226 TM5 L => A N/A N/A Blaker M et al (2000)
gasr_human 5.47x47 227 TM5 F => A N/A N/A Blaker M et al (2000)
gasr_human 6.48x48 346 TM6 W => A N/A N/A Blaker M et al (2000)
gasr_human 6.51x51 349 TM6 V => A N/A N/A Blaker M et al (2000)
gasr_human 6.52x52 350 TM6 Y => A N/A N/A Blaker M et al (2000)
gasr_human 6.55x55 353 TM6 N => L N/A N/A Blaker M et al (2000)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Blaker M et al (2000)
gasr_human 7.42x41 379 TM7 S => A N/A N/A Blaker M et al (2000)
gasr_human 1.35x35 57 TM1 R => A N/A N/A Langer I et al (2005)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Kopin AS et al (1995)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Langer I et al (2005)
gasr_human 1.39x39 61 TM1 Y => A N/A N/A Blaker M et al (2000)
gasr_human 12.50x50 85 ICL1 L => M N/A N/A Wu SV et al (1999)
gasr_human 2.57x56 107 TM2 C => A N/A N/A Blaker M et al (2000)
gasr_human 2.60x59 110 TM2 F => A N/A N/A Blaker M et al (2000)
gasr_human 2.61x60 111 TM2 T => A N/A N/A Blaker M et al (2000)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 23.50x50 120 ECL1 F => A N/A N/A Langer I et al (2005)
gasr_human 3.29x29 131 TM3 S => A N/A N/A Blaker M et al (2000)
gasr_human 3.29x29 131 TM3 S => T N/A N/A Kopin AS et al (1995)
gasr_human 3.32x32 134 TM3 M => L N/A N/A Dong M et al (2005)
gasr_human 3.33x33 135 TM3 G => A N/A N/A Blaker M et al (2000)
gasr_human 3.36x36 138 TM3 V => A N/A N/A Blaker M et al (2000)
gasr_human 4.57x57 186 TM4 M => A N/A N/A Blaker M et al (2000)
gasr_human 4.60x61 189 TM4 Y => A N/A N/A Langer I et al (2005)
gasr_human 4.60x61 189 TM4 Y => F N/A N/A Langer I et al (2005)
gasr_human 4.64x65 193 TM4 T => A N/A N/A Blaker M et al (2000)
gasr_human 45.51x51 206 ECL2 V => M N/A N/A Langer I et al (2005)
gasr_human 45.52x52 207 ECL2 H => A N/A N/A Langer I et al (2005)
gasr_human 5.39x40 219 TM5 S => A N/A N/A Blaker M et al (2000)
gasr_human 5.39x40 219 TM5 S => H N/A N/A Kopin AS et al (1995)
gasr_human 5.43x44 223 TM5 L => A N/A N/A Blaker M et al (2000)
gasr_human 5.47x47 227 TM5 F => A N/A N/A Blaker M et al (2000)
gasr_human 5.54x54 234 TM5 M => I N/A N/A Langer I et al (2005)
gasr_human 6.48x48 346 TM6 W => A N/A N/A Blaker M et al (2000)
gasr_human 6.51x51 349 TM6 V => A N/A N/A Blaker M et al (2000)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Kopin AS et al (1995)
gasr_human 6.52x52 350 TM6 Y => A N/A N/A Blaker M et al (2000)
gasr_human 6.52x52 350 TM6 Y => F N/A N/A Kopin AS et al (1995)
gasr_human 6.55x55 353 TM6 N => A N/A N/A Langer I et al (2005)
gasr_human 6.55x55 353 TM6 N => L N/A N/A Blaker M et al (2000)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Blaker M et al (2000)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 6.58x58 356 TM6 R => A N/A N/A Langer I et al (2005)
gasr_human 6.58x58 356 TM6 R => D N/A N/A Langer I et al (2005)
gasr_human 6.58x58 356 TM6 R => H N/A N/A Langer I et al (2005)
gasr_human 6.58x58 356 TM6 R => I N/A N/A Langer I et al (2005)
gasr_human 6.58x58 356 TM6 R => K N/A N/A Langer I et al (2005)
gasr_human 7.39x38 376 TM7 H => A N/A N/A Gouldson P et al (1999)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Gouldson P et al (1999)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Silvente-Poirot S et al (1998)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Langer I et al (2005)
gasr_human 7.42x41 379 TM7 S => A N/A N/A Blaker M et al (2000)
gasr_human 7.42x41 379 TM7 S => A N/A N/A Blaker M et al (2000)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Blaker M et al (2000)
gasr_human 6.55x55 353 TM6 N => L N/A N/A Blaker M et al (2000)
gasr_human 6.52x52 350 TM6 Y => A N/A N/A Blaker M et al (2000)
gasr_human 6.51x51 349 TM6 V => A N/A N/A Blaker M et al (2000)
gasr_human 6.48x48 346 TM6 W => A N/A N/A Blaker M et al (2000)
gasr_human 5.47x47 227 TM5 F => A N/A N/A Blaker M et al (2000)
gasr_human 5.46x461 226 TM5 L => A N/A N/A Blaker M et al (2000)
gasr_human 5.43x44 223 TM5 L => A N/A N/A Blaker M et al (2000)
gasr_human 5.39x40 219 TM5 S => A N/A N/A Blaker M et al (2000)
gasr_human 4.64x65 193 TM4 T => A N/A N/A Blaker M et al (2000)
gasr_human 3.36x36 138 TM3 V => A N/A N/A Blaker M et al (2000)
gasr_human 4.57x57 186 TM4 M => A N/A N/A Blaker M et al (2000)
gasr_human 3.33x33 135 TM3 G => A N/A N/A Blaker M et al (2000)
gasr_human 3.29x29 131 TM3 S => A N/A N/A Blaker M et al (2000)
gasr_human 2.61x60 111 TM2 T => A N/A N/A Blaker M et al (2000)
gasr_human 2.57x56 107 TM2 C => A N/A N/A Blaker M et al (2000)
gasr_human 2.60x59 110 TM2 F => A N/A N/A Blaker M et al (2000)
gasr_human 1.39x39 61 TM1 Y => A N/A N/A Blaker M et al (2000)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 6.52x52 350 TM6 Y => F N/A N/A Kopin AS et al (1995)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => H N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => Q N/A N/A Kopin AS et al (1995)
gasr_human 3.29x29 131 TM3 S => T N/A N/A Kopin AS et al (1995)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Kopin AS et al (1995)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => H N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => Q N/A N/A Kopin AS et al (1995)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Kopin AS et al (1995)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => H N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => Q N/A N/A Kopin AS et al (1995)
gasr_human 3.29x29 131 TM3 S => T N/A N/A Kopin AS et al (1995)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Kopin AS et al (1995)
gasr_human 7.39x38 376 TM7 H => L N/A N/A Kopin AS et al (1995)
gasr_human 6.56x56 354 TM6 T => A N/A N/A Kopin AS et al (1995)
gasr_human 6.51x51 349 TM6 V => I N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => I N/A N/A Kopin AS et al (1995)
gasr_human 5.39x40 219 TM5 S => Q N/A N/A Kopin AS et al (1995)
gasr_human 3.29x29 131 TM3 S => T N/A N/A Kopin AS et al (1995)
gasr_human 2.61x60 111 TM2 T => N N/A N/A Kopin AS et al (1995)
gasr_human 1.35x35 57 TM1 R => Q N/A N/A Kopin AS et al (1995)
gasr_human 5.73x73 253 TM5 G => E N/A N/A Brockhoff A et al (2010)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 R R L R ICL1ECL1 T F I F ECL1ICL2 P L Q A R V W Q ICL2ECL2 V V Q P V G P R V L Q C V H R W P ECL2ICL3 S D S Q S R V R N Q G G L P G A V H Q N G R C R P E T G A V G E D S D G C Y V Q L P R S R P A L E L T A L T A P G P G S G S R P T ICL3ECL3 P G A H R A L S ECL3N-term M E L L K L N R S V Q G T G P G P G A S L C R P G A P L L N S S S V G N L S C E P P R I R G A G T R E N-termC-term A R C C P R P P R A R P R A L P D E D P P T P S I A S L S R L S Y T T I S T L G P G C-term L E L A I R I T L Y A V I F L M S V G G N M L I I V V L G L S T V T N A F L L S L A V S D L L L A V A C M P F T L L P N L M G G T V I C K A V S Y L M G V S V S V S T L S L V A I A L E R Y S A I C R T R S H A A R V I V A T W L L S G L L M V P Y P V Y T S A R V R Q T W S V L L L L L L F F I P G V V M A V A Y G L I S R E L Y L G L R F D G D S D Q A K L L A K K R V V R M L L V I V V L F F L C W L P V Y S A N T W R A F D G G A P I S F I H L L S Y A S A C V N P L V Y C F M H R R C L E F R Q A T C
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
M N G G V S M L F I V A Y L T I R I A L 1 L S L A V S D L L L A A V C M P F T L L P 2 A V L S L T S V S V S V G M L Y S V A K 3 A A R V I V A T W L L S G L L M V P Y 4 Y A V A M V V G P I F F L L L L L L V S W 5 L V I V V L F F L C W L P V Y S A N T W 6 L P N V C A S A Y S L L H I F S I P A 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
CCK2 receptor
TM1
1x34 1.34x34 I56
1x35 1.35x35 R57
1x37 1.37x37 T59
1x39 1.39x39 Y61
1x41 1.41x41 V63
1x51 1.51x51 M73
1x58 1.58x58 G80
1x60 1.60x60 S82
TM2
2x41 2.41x41 A91
2x56 2.57x56 C107
2x59 2.60x59 F110
2x60 2.61x60 T111
TM3
3x27 3.27x27 A129
3x28 3.28x28 V130
3x29 3.29x29 S131
3x31 3.31x31 L133
3x32 3.32x32 M134
3x33 3.33x33 G135
3x34 3.34x34 V136
3x36 3.36x36 V138
3x47 3.47x47 A149
TM4
4x47 4.47x47 V176
4x51 4.51x51 L180
4x57 4.57x57 M186
4x61 4.60x61 Y189
4x65 4.64x65 T193
TM5
5x40 5.39x40 S219
5x44 5.43x44 L223
5x46 5.45x46 L225
5x461 5.46x461 L226
5x47 5.47x47 F227
5x49 5.49x49 I229
5x54 5.54x54 M234
5x55 5.55x55 A235
5x73 5.73x73 G253
TM6
6x48 6.48x48 W346
6x49 6.49x49 L347
6x51 6.51x51 V349
6x52 6.52x52 Y350
6x55 6.55x55 N353
6x56 6.56x56 T354
6x58 6.58x58 R356
TM7
7x32 7.33x32 A370
7x38 7.39x38 H376
7x41 7.42x41 S379
7x43 7.44x43 A381
7x46 7.46x46 A383