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STRUCTURE
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RECEPTOR
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ARRESTIN
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OTHER PROTEINS
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STRUCTURE LIGAND
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REFERENCE
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PDB
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Method | Resolution |
UniProt
|
Gene | IUPHAR | Receptor family | Class | Species | Fam. | Arrestin | Species | Note | % of Seq | Receptor fusion | Antibodies | Other | Name | Type | Function | Authors | Reference | PDB Date | ||
| 5DGY | X-ray | 7.7 | OPSD | RHO | Rhodopsin | Opsin (sight) | A (Rhodopsin) | Human | Visual | S-arrestin | Mouse | Rhodopsin C-term fusion, 15aa linker, 3A muts | 86 | T4-Lysozyme | - | - | - | None | - | Zhou XE, Gao X, Barty A, Kang Y, He Y, Liu W, Ishchenko A, White TA, Yefanov O, Han GW, Xu Q, de Waal PW, Suino-Powell KM, Boutet S, Williams GJ, Wang M, Li D, Caffrey M, Chapman HN, Spence JC, Fromme P, Weierstall U, Stevens RC, Cherezov V, Melcher K, Xu HE | 10.1038/SDATA.2016.21 | 2016-03-23 | 58504 | |
| 8WRZ | Cryo-EM | 3.6 | CNR1 | CNR1 | CB1 | Cannabinoid | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 84 | BRIL | - | - |
AM841
pubchem
gtoplig
chembl_ligand
V2Rpp (phosphorylated Vasopressin V2 receptor C-terminal tail) |
Small molecule Peptide |
Agonist | Wang Y, Wu L, Wang T, Liu J, Li F, Jiang L, Fan Z, Yu Y, Chen N, Sun Q, Tan Q, Hua T, Liu ZJ | 10.1093/PROCEL/PWAD055 | 2024-02-28 | 58438 | |
| 6U1N | Cryo-EM | 4.0 | ACM2 | CHRM2 | M2 | Acetylcholine (muscarinic) | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Rat | M2R-V2Rpp fusion stabilizes β-arr1 binding | 86 | - | - | - |
iperoxo
pubchem
gtoplig
chembl_ligand
LY2119620 pubchem gtoplig chembl_ligand |
Small molecule Small molecule |
Agonist PAM |
Staus DP, Hu H, Robertson MJ, Kleinhenz ALW, Wingler LM, Capel WD, Latorraca NR, Lefkowitz RJ, Skiniotis G | 10.1038/S41586-020-1954-0 | 2020-02-26 | 58440 | |
| 6UP7 | Cryo-EM | 4.2 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Human β-arr1 ΔCT (truncated at res 382) | 83 | - | - | - |
NTS8–13
pubchem
PIO pubchem |
Peptide Small molecule |
Agonist PAM |
Huang W, Masureel M, Qu Q, Janetzko J, Inoue A, Kato HE, Robertson MJ, Nguyen KC, Glenn JS, Skiniotis G, Kobilka BK | 10.1038/S41586-020-1953-1 | 2020-02-26 | 58438 | |
| 8JRV | Cryo-EM | 3.3 | GLR | GCGR | glucagon | Glucagon | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Bovine | Cys-free β-arr1 (7 Cys muts), R169E, scFv30 | 85 | - | Nanobody 32 | - |
Glucagon
pubchem
|
Small molecule | Agonist | Chen K, Zhang C, Lin S, Yan X, Cai H, Yi C, Ma L, Chu X, Liu Y, Zhu Y, Han S, Zhao Q, Wu B | 10.1038/S41586-023-06420-X | 2023-08-16 | 58441 | |
| 8ZYU | Cryo-EM | 2.7 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Active variant, Δ382 trunc, no autoinhibition | 87 | BRIL | - | - |
NTS8–13
pubchem
SBI-553 pubchem gtoplig chembl_ligand |
Peptide Small molecule |
Agonist Allosteric agonist |
Sun D, Li X, Yuan Q, Wang Y, Shi P, Zhang H, Wang T, Sun W, Ling S, Liu Y, Lai J, Xie W, Yin W, Liu L, Xu HE, Tian C | 10.1038/S41422-025-01095-7 | 2025-04-16 | 58438 | |
| 9KUV | Cryo-EM | 3.2 | APJ | APLNR | apelin | Apelin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Cys-free β-arr1, R169E mut, C-term scFv30 fusion | 139 | BRIL | - | V2R C-tail |
cmpd644
pubchem
|
Small molecule | Agonist | - | - | 2025-09-17 | 58438 | |
| 9KUW | Cryo-EM | 3.5 | APJ | APLNR | apelin | Apelin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Cys-deficient β-arr, R169E, scFv30 fusion | 139 | BRIL | - | - |
cmpd644
pubchem
|
Small molecule | Agonist | - | - | 2025-09-17 | 58438 | |
| 9KUX | Cryo-EM | 3.6 | APJ | APLNR | apelin | Apelin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Cys-free β-arr1, C-term scFv30 fusion | 138 | BRIL | - | - |
cmpd644
pubchem
|
Small molecule | Agonist | - | - | 2025-09-17 | 58438 | |
| 9UCO | Cryo-EM | 3.6 | AGRE1 | Adgre1 | ADGRE1 | ADGRE | B2 (Adhesion) | Mouse | Beta | Beta-arrestin-1 | Bovine | 2 β-arr1 copies bind the receptor dimer | 83 | - | - | - |
Stalk peptide
|
Peptide | Agonist | - | - | 2026-04-08 | 58441 | |
| 9L8L | Cryo-EM | 3.2 | ADRB2 | ADRB2 | β2 | Adrenoceptors | A (Rhodopsin) | Human | Gs | s | Bovine | Gs heterotrimer: bovine Gα, rat Gβ, bovine Gγ | 58 | - | - | - |
ATAZANAVIR
chembl_ligand
pubchem
drugbank
CHEMBL1615159 chembl_ligand pubchem |
Small molecule Small molecule |
Ago-PAM Agonist |
He G, Sun Q, Xu X, Kong F, Zhang S, Ye K, Sun X, Lin B, Chen X, Yan C, Liu X | 10.1016/J.CELL.2025.12.023 | 2025-12-31 | 58438 | |
| 9LZ1 | Cryo-EM | 3.2 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Bovine | - | 83 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-11 | 58441 | |
| 9UYN | Cryo-EM | 2.9 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 82 | - | Nanobody 32 | - |
Palmitoleic Acid
pubchem
drugbank
|
Small molecule | Allosteric agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58438 | |
| 9LXP | Cryo-EM | 3.2 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Human | - | 83 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-04 | 58438 | |
| 5W0P | X-ray | 3.0 | OPSD | RHO | Rhodopsin | Opsin (sight) | A (Rhodopsin) | Human | Visual | S-arrestin | Mouse | Visual arrestin fused to receptor C-term | 90 | T4-Lysozyme | - | - | - | None | - | Zhou XE, He Y, de Waal PW, Gao X, Kang Y, Van Eps N, Yin Y, Pal K, Goswami D, White TA, Barty A, Latorraca NR, Chapman HN, Hubbell WL, Dror RO, Stevens RC, Cherezov V, Gurevich VV, Griffin PR, Ernst OP, Melcher K, Xu HE | 10.1016/J.CELL.2017.07.002 | 2017-08-09 | 58504 | |
| 4PXF | X-ray | 2.8 | OPSD | RHO | Rhodopsin | Opsin (sight) | A (Rhodopsin) | Bovine | Visual | S-arrestin | Bovine | ArrFL-1 peptide: rod arrestin finger loop 67-77 | 2 | - | - | - | - | None | - | Szczepek M, Beyriere F, Hofmann KP, Elgeti M, Kazmin R, Rose A, Bartl FJ, von Stetten D, Heck M, Sommer ME, Hildebrand PW, Scheerer P | 10.1038/NCOMMS5801 | 2014-09-17 | 58515 | |
| 4ZWJ | X-ray | 3.3 | OPSD | RHO | Rhodopsin | Opsin (sight) | A (Rhodopsin) | Human | Visual | S-arrestin | Mouse | - | 86 | T4-Lysozyme | - | - | - | None | - | Kang Y, Zhou XE, Gao X, He Y, Liu W, Ishchenko A, Barty A, White TA, Yefanov O, Han GW, Xu Q, de Waal PW, Ke J, Tan MH, Zhang C, Moeller A, West GM, Pascal BD, Van Eps N, Caro LN, Vishnivetskiy SA, Lee RJ, Suino-Powell KM, Gu X, Pal K, Ma J, Zhi X, Boutet S, Williams GJ, Messerschmidt M, Gati C, Zatsepin NA, Wang D, James D, Basu S, Roy-Chowdhury S, Conrad CE, Coe J, Liu H, Lisova S, Kupitz C, Grotjohann I, Fromme R, Jiang Y, Tan M, Yang H, Li J, Wang M, Zheng Z, Li D, Howe N, Zhao Y, Standfuss J, Diederichs K, Dong Y, Potter CS, Carragher B, Caffrey M, Jiang H, Chapman HN, Spence JC, Fromme P, Weierstall U, Ernst OP, Katritch V, Gurevich VV, Griffin PR, Hubbell WL, Stevens RC, Cherezov V, Melcher K, Xu HE | 10.1038/NATURE14656 | 2015-07-29 | 58504 | |
| 6TKO | Cryo-EM | 3.3 | ADRB1 | ADRB1 | β1 | Adrenoceptors | A (Rhodopsin) | Wild turkey | Beta | Beta-arrestin-1 | Human | β-arr1 (arrestin2), L68C+R169E muts | 82 | - | - | - |
ARFORMOTEROL
chembl_ligand
pubchem
drugbank
drug_central
pubchem
drugbank
|
Small molecule | Agonist | Lee Y, Warne T, Nehme R, Pandey S, Dwivedi-Agnihotri H, Chaturvedi M, Edwards PC, Garcia-Nafria J, Leslie AGW, Shukla AK, Tate CG | 10.1038/S41586-020-2419-1 | 2020-06-17 | 58438 | |
| 6PWC | Cryo-EM | 4.9 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 84 | - | - | - |
NTS8–13
pubchem
|
Peptide | Agonist | Yin W, Li Z, Jin M, Yin YL, de Waal PW, Pal K, Yin Y, Gao X, He Y, Gao J, Wang X, Zhang Y, Zhou H, Melcher K, Jiang Y, Cong Y, Edward Zhou X, Yu X, Eric Xu H | 10.1038/S41422-019-0256-2 | 2019-12-04 | 58438 | |
| 7R0C | Cryo-EM | 4.7 | V2R | AVPR2 | V2 | Vasopressin and oxytocin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Human β-arr1 (res 6-365), ΔCT at 382 | 84 | - | - | - |
vasopressin (Human)
pubchem
gtoplig
chembl_ligand
drugbank
drug_central
uniprot
uniprot
uniprot
pubchem
pubchem
|
Peptide | Agonist | Bous J, Fouillen A, Orcel H, Trapani S, Cong X, Fontanel S, Saint-Paul J, Lai-Kee-Him J, Urbach S, Sibille N, Sounier R, Granier S, Mouillac B, Bron P | 10.1126/SCIADV.ABO7761 | 2022-09-14 | 58438 | |
| 7SRS | Cryo-EM | 3.3 | 5HT2B | HTR2B | 5-HT2B | 5-Hydroxytryptamine | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Isoform 1B, R169E, truncated to res 1-368 | 85 | BRIL | - | - |
(+)-LSD
pubchem
gtoplig
pubchem
gtoplig
chembl_ligand
drugbank
drug_central
|
Small molecule | Agonist (partial) | Cao C, Barros-Alvarez X, Zhang S, Kim K, Damgen MA, Panova O, Suomivuori CM, Fay JF, Zhong X, Krumm BE, Gumpper RH, Seven AB, Robertson MJ, Krogan NJ, Huttenhain R, Nichols DE, Dror RO, Skiniotis G, Roth BL | 10.1016/J.NEURON.2022.08.006 | 2022-09-21 | 58438 | |
| 8JRU | Cryo-EM | 3.5 | GLR | GCGR | glucagon | Glucagon | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Bovine | Cys-free bo β-arr1, R169E, scFv30 C-term swap | 83 | - | Nanobody 32 | - | - | None | - | Chen K, Zhang C, Lin S, Yan X, Cai H, Yi C, Ma L, Chu X, Liu Y, Zhu Y, Han S, Zhao Q, Wu B | 10.1038/S41586-023-06420-X | 2023-08-16 | 58441 | |
| 9M0D | Cryo-EM | 3.4 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Active β-arr variant truncated at res 382 | 86 | BRIL | - | - | - | None | - | - | - | 2025-04-09 | 58438 | |
| 8WU1 | Cryo-EM | 3.2 | CNR1 | CNR1 | CB1 | Cannabinoid | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Bovine | - | 86 | - | - | - |
MDMB-Fubinaca
pubchem
gtoplig
|
Small molecule | Agonist | Liao YY, Zhang H, Shen Q, Cai C, Ding Y, Shen DD, Guo J, Qin J, Dong Y, Zhang Y, Li XM | 10.1016/J.CELL.2023.11.017 | 2024-03-20 | 58441 | |
| 9E82 | Cryo-EM | 3.4 | ACKR3 | ACKR3 | ACKR3 | Chemokine | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Bovine | - | 81 | - | - | - |
SDF-1-beta(3-72)
|
Peptide | Agonist | Chen Q, Schafer CT, Mukherjee S, Wang K, Gustavsson M, Fuller JR, Tepper K, Lamme TD, Aydin Y, Agrawal P, Terashi G, Yao XQ, Kihara D, Kossiakoff AA, Handel TM, Tesmer JJG | 10.1038/S41586-025-09024-9 | 2025-04-02 | 58441 | |
| 9IJS | Cryo-EM | 3.6 | GPR52 | GPR52 | GPR52 | Orphan | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 84 | - | - | - | - | None | - | Lin X, Wei X, Pu N, Wang L, Zhang Z, Li C, Yue Y, Liu J, Tan Q, Sun Q, Xu F | 10.1038/S41422-025-01165-W | 2025-09-03 | 58438 | |
| 9LXR | Cryo-EM | 3.1 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Human | - | 83 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2025-09-10 | 58438 | |
| 8ZYT | Cryo-EM | 2.7 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Active β-arr, Δ382 trunc, no autoinhibition | 86 | BRIL | - | - |
NTS8–13
pubchem
SBI-553 pubchem gtoplig chembl_ligand |
Peptide Small molecule |
Agonist Allosteric agonist |
- | - | 2025-04-09 | 58438 | |
| 8ZYY | Cryo-EM | 2.8 | NTR1 | NTSR1 | NTS1 | Neurotensin | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | Truncated at res 382, autoinhibition removed | 86 | BRIL | - | - |
NTS8–13
pubchem
SBI-553 pubchem gtoplig chembl_ligand |
Peptide Small molecule |
Agonist Allosteric agonist |
- | - | 2025-04-09 | 58438 | |
| 9II2 | Cryo-EM | 3.7 | GRM3 | GRM3 | mGlu3 | Metabotropic glutamate | C (Glutamate) | Human | Beta | Beta-arrestin-1 | Human | Active Cys-free β-arr1(1-376) R169E+scFv30 | 83 | - | - | - |
L-glutamic acid
pubchem
gtoplig
chembl_ligand
drugbank
drug_central
chembl_ligand
pubchem
pubchem
drugbank
|
Small molecule | Agonist | Wen T, Du M, Lu Y, Jia N, Lu X, Liu N, Chang S, Zhang X, Shen Y, Yang X | 10.1038/S41589-025-01858-8 | 2025-03-05 | 58438 | |
| 9II3 | Cryo-EM | 3.9 | GRM3 | GRM3 | mGlu3 | Metabotropic glutamate | C (Glutamate) | Human | Beta | Beta-arrestin-1 | Human | Active Cys-free β-arr1(1-376), R169E mut | 83 | - | - | - |
L-glutamic acid
pubchem
gtoplig
chembl_ligand
drugbank
drug_central
chembl_ligand
pubchem
pubchem
drugbank
|
Small molecule | Agonist | Wen T, Du M, Lu Y, Jia N, Lu X, Liu N, Chang S, Zhang X, Shen Y, Yang X | 10.1038/S41589-025-01858-8 | 2025-03-05 | 58438 | |
| 9IJR | Cryo-EM | 3.9 | GPR52 | GPR52 | GPR52 | Orphan | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | β-arr1 binds GPR52 via ICL1/H8 side engagement | 84 | - | - | - |
derivative 17 [Nakahata et al., 2018]
pubchem
gtoplig
chembl_ligand
|
Small molecule | Agonist | Lin X, Wei X, Pu N, Wang L, Zhang Z, Li C, Yue Y, Liu J, Tan Q, Sun Q, Xu F | 10.1038/S41422-025-01165-W | 2025-09-03 | 58438 | |
| 9LY2 | Cryo-EM | 3.1 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Human | - | 80 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-04 | 58438 | |
| 9LY3 | Cryo-EM | 3.4 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Human | Full-length β-arrestin-1 | 80 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-04 | 58438 | |
| 9LZ0 | Cryo-EM | 3.8 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Bovine | - | 83 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-18 | 58441 | |
| 9LZ2 | Cryo-EM | 3.0 | PTH1R | PTH1R | PTH1 | Parathyroid hormone | B1 (Secretin) | Human | Beta | Beta-arrestin-1 | Bovine | β-arr1 stabilized by Fab30 | 83 | - | - | - |
Long-acting parathyroid hormone analog
pubchem
|
Peptide | Agonist | - | - | 2026-03-11 | 58441 | |
| 9MBA | Cryo-EM | 3.1 | GRM8 | GRM8 | mGlu8 | Metabotropic glutamate | C (Glutamate) | Human | Beta | Beta-arrestin-1 | Human | Truncated at 377, R169E, no autoinhibition | 79 | - | - | - |
L-glutamic acid
pubchem
gtoplig
chembl_ligand
drugbank
drug_central
chembl_ligand
pubchem
pubchem
drugbank
|
Small molecule | Agonist | Zhao J, Deng Y, Xu Z, Xu C, Zhao C, Li Z, Sun H, Tian X, Song Y, Cimadevila M, Wang H, Liu Y, Zhang X, Chen Y, Sun S, Yong X, Su L, He Y, Zhong Y, Yang H, Pin JP, Yan W, Shao Z, Liu J | 10.1016/J.MOLCEL.2025.08.019 | 2025-10-01 | 58438 | |
| 9UYL | Cryo-EM | 3.3 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 77 | - | Nanobody 32 | - |
Chemerin
|
Protein | Agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58438 | |
| 9UYH | Cryo-EM | 3.3 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 81 | - | Nanobody 32 | - |
Chemerin
|
Protein | Agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58438 | |
| 9UYI | Cryo-EM | 3.2 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | β-arr1 stabilized by Nb32 and scFv30 | 79 | - | Nanobody 32 | - |
Chemerin
|
Protein | Agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58438 | |
| 9UYJ | Cryo-EM | 3.3 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 78 | - | Nanobody 32 | - |
Chemerin
|
Protein | Agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58438 | |
| 9UYM | Cryo-EM | 3.5 | CML2 | CMKLR2 | chemerin 2 | Chemerin receptor | A (Rhodopsin) | Human | Beta | Beta-arrestin-2 | Human | β-arr2 tail swap (H350-F376→β-arr1) for scFv30 | 77 | - | Nanobody 32 | - |
Chemerin
|
Protein | Agonist | Cai H, Lin X, Zhao L, He M, Yu J, Zhang B, Ma Y, Chang X, Tang Y, Luo T, Jiang J, Ma M, Song W, Ma L, Chu X, Yi C, Chen K, Han S, Xie C, Shui W, Zhao Q, Zhu Y, Wu B | 10.1126/SCIENCE.ADT8794 | 2025-11-19 | 58461 | |
| 9WSV | Cryo-EM | 2.8 | OPRM | Oprm1 | μ | Opioid | A (Rhodopsin) | Mouse | Beta | Beta-arrestin-1 | Bovine | Active bo β-arr1: R169E+I386A/V387A/F388A | 84 | - | - | - |
DAMGO
pubchem
gtoplig
chembl_ligand
pubchem
|
Peptide | Agonist | Zhang H, Wang X, Xi K, Shen Q, Xue J, Zhu Y, Zang SK, Yu T, Shen DD, Guo J, Chen LN, Ji SY, Qin J, Dong Y, Zhao M, Yang M, Wu H, Yang G, Zhang Y | 10.1038/S41422-025-01191-8 | 2025-11-26 | 58441 | |
| 9WSX | Cryo-EM | 2.8 | OPRM | Oprm1 | μ | Opioid | A (Rhodopsin) | Mouse | Beta | Beta-arrestin-1 | Bovine | Bo β-arr1 Δ394, R169E+I386A/V387A/F388A muts | 84 | - | - | - |
endomorphin-1 (Human)
pubchem
gtoplig
chembl_ligand
|
Peptide | Agonist | Zhang H, Wang X, Xi K, Shen Q, Xue J, Zhu Y, Zang SK, Yu T, Shen DD, Guo J, Chen LN, Ji SY, Qin J, Dong Y, Zhao M, Yang M, Wu H, Yang G, Zhang Y | 10.1038/S41422-025-01191-8 | 2025-11-26 | 58441 | |
| 9ZZO | Cryo-EM | 2.6 | OPRK | OPRK1 | κ | Opioid | A (Rhodopsin) | Human | Beta | Beta-arrestin-1 | Human | - | 84 | - | Nanobody 32 | - |
CHEMBL5431513
chembl_ligand
pubchem
|
Small molecule | Agonist | Han J, Fine EJ, Jiang Q, Zhuang Y, Suomivuori CM, Chen ZW, Denn E, Whiddon K, Li K, Evers AS, Fuller J, Carter J, Fay JF, Chen M, Dror RO, Che T | 10.1038/S41467-026-73968-3 | 2026-06-17 | 58438 | |
| 1G4M | X-ray | 1.9 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | - | - | - | - | Han M, Gurevich VV, Vishnivetskiy SA, Sigler PB, Schubert C | 11566136 | 2001-10-03 | 58441 | |
| 1G4R | X-ray | 2.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | - | - | - | - | Han M, Gurevich VV, Vishnivetskiy SA, Sigler PB, Schubert C | 11566136 | 2001-10-03 | 58441 | |
| 1JSY | X-ray | 2.9 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | - | - | - | - | Milano SK, Pace HC, Kim YM, Brenner C, Benovic JL | 11876640 | 2002-03-27 | 58441 | |
| 1ZSH | X-ray | 2.9 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | - | - | - | - | Milano SK, Kim YM, Stefano FP, Benovic JL, Brenner C | 16439357 | 2006-01-31 | 58441 | |
| 2WTR | X-ray | 2.9 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | - | - | - | - | - | - | 2009-09-29 | 58441 | |
| 3GC3 | X-ray | 2.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | Clathrin heavy chain 1 | - | - | - | Kang DS, Kern RC, Puthenveedu MA, von Zastrow M, Williams JC, Benovic JL | 19710023 | 2009-08-25 | 58441 | |
| 3GD1 | X-ray | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | - | Clathrin heavy chain 1 clathrin |
- | - | - | Kang DS, Kern RC, Puthenveedu MA, von Zastrow M, Williams JC, Benovic JL | 19710023 | 2009-08-25 | 58441 | |
| 6NI2 | Cryo-EM | 4.0 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Nanobody 32 Fab30 Heavy Chain Fab30 Light Chain |
Vasopressin V2 receptor | - | - | - | Nguyen AH, Thomsen ARB, Cahill TJ 3rd, Huang R, Huang LY, Marcink T, Clarke OB, Heissel S, Masoudi A, Ben-Hail D, Samaan F, Dandey VP, Tan YZ, Hong C, Mahoney JP, Triest S, Little J 4th, Chen X, Sunahara R, Steyaert J, Molina H, Yu Z, des Georges A, Lefkowitz RJ | 31740855 | 2019-11-20 | 58441 | |
| 7DF9 | X-ray | 3.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 Light Chain Fab30 Heavy Chain |
Vasopressin V2 receptor phosphopeptide | - | - | - | He QT, Xiao P, Huang SM, Jia YL, Zhu ZL, Lin JY, Yang F, Tao XN, Zhao RJ, Gao FY, Niu XG, Xiao KH, Wang J, Jin C, Sun JP, Yu X | 33888704 | 2021-07-28 | 58441 | |
| 7DFA | X-ray | 2.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
VaRpp-4 | - | - | - | He QT, Xiao P, Huang SM, Jia YL, Zhu ZL, Lin JY, Yang F, Tao XN, Zhao RJ, Gao FY, Niu XG, Xiao KH, Wang J, Jin C, Sun JP, Yu X | 33888704 | 2021-07-28 | 58441 | |
| 7DFB | X-ray | 3.3 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 Light Chain Fab30 Heavy Chain |
V2Rpp-6-7 | - | - | - | He QT, Xiao P, Huang SM, Jia YL, Zhu ZL, Lin JY, Yang F, Tao XN, Zhao RJ, Gao FY, Niu XG, Xiao KH, Wang J, Jin C, Sun JP, Yu X | 33888704 | 2021-07-28 | 58441 | |
| 7DFC | X-ray | 2.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 Light Chain Fab30 Heavy Chain |
V2Rpp-3 | - | - | - | He QT, Xiao P, Huang SM, Jia YL, Zhu ZL, Lin JY, Yang F, Tao XN, Zhao RJ, Gao FY, Niu XG, Xiao KH, Wang J, Jin C, Sun JP, Yu X | 33888704 | 2021-07-28 | 58441 | |
| 8J97 | Cryo-EM | 3.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Muscarinic acetylcholine receptor M2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58441 | |
| 8JAF | Cryo-EM | 3.1 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab30 heavy chain Fab30 light chain |
Muscarinic acetylcholine receptor M2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58441 | |
| 8TII | Cryo-EM | 3.0 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Bovine | - | - | - | Fab7 heavy chain Fab7 light chain anti-Fab nanobody |
Atypical chemokine receptor 3 | - | - | - | Chen Q, Schafer CT, Mukherjee S, Wang K, Gustavsson M, Fuller JR, Tepper K, Lamme TD, Aydin Y, Agrawal P, Terashi G, Yao XQ, Kihara D, Kossiakoff AA, Handel TM, Tesmer JJG | 40399676 | 2025-01-22 | 58441 | |
| 4JQI | X-ray | 2.6 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 heavy chain Fab30 light chain |
Vasopressin V2 receptor phosphopeptide | - | - | - | Shukla AK, Manglik A, Kruse AC, Xiao K, Reis RI, Tseng WC, Staus DP, Hilger D, Uysal S, Huang LY, Paduch M, Tripathi-Shukla P, Koide A, Koide S, Weis WI, Kossiakoff AA, Kobilka BK, Lefkowitz RJ | 23604254 | 2013-04-17 | 58440 | |
| 6KL7 | X-ray | 2.8 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | - | - | - | - | - | Kang H, Yang HS, Ki AY, Ko SB, Kim KW, Shim CY, Kim K, Choi HJ, Chung KY | 31948726 | 2020-01-29 | 58440 | |
| 8GO8 | Cryo-EM | 3.4 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 heavy chain Fab30 light chain |
C5a anaphylatoxin chemotactic receptor 1 | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58440 | |
| 8GP3 | Cryo-EM | 4.8 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C-X-C chemokine receptor type 4 | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58440 | |
| 8HST | X-ray | 2.7 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | - | - | - | - | - | Yun Y, Yoon HJ, Jeong Y, Choi Y, Jang S, Chung KY, Lee HH | 37399373 | 2023-07-19 | 58440 | |
| 8HSV | X-ray | 3.0 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | - | peptide from E3 ubiquitin-protein ligase Mdm2 | - | - | - | Yun Y, Yoon HJ, Jeong Y, Choi Y, Jang S, Chung KY, Lee HH | 37399373 | 2023-07-19 | 58440 | |
| 8I0Q | Cryo-EM | 4.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C-X-C chemokine receptor type 4 | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58440 | |
| 8J8Z | Cryo-EM | 3.4 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Atypical chemokine receptor 2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58440 | |
| 8JA3 | Cryo-EM | 3.9 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 heavy chain Fab30 light chain |
C3a anaphylatoxin chemotactic receptor | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58440 | |
| 9BT8 | Cryo-EM | 3.3 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Antibody fragment Fab30 Nanobody 32 Antibody fragment Fab30 |
Proto-oncogene tyrosine-protein kinase Src heavy chain Vasopressin V2 receptor light chain |
- | - | - | Pakharukova N, Thomas BN, Bansia H, Li L, Bassford DK, Abzalimov RR, Kim J, Kahsai AW, Pani B, Xiao K, Ochakovski R, Liu S, Zhang X, Ahn S, des Georges A, Lefkowitz RJ | 41720803 | 2024-11-13 | 58440 | |
| 9CX3 | Cryo-EM | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Nanobody 32 Antibody fragment Fab30 Antibody fragment Fab30 |
Proto-oncogene tyrosine-protein kinase Src heavy chain Vasopressin V2 receptor light chain |
- | - | - | Pakharukova N, Thomas BN, Bansia H, Li L, Bassford DK, Abzalimov RR, Kim J, Kahsai AW, Pani B, Xiao K, Ochakovski R, Liu S, Zhang X, Ahn S, des Georges A, Lefkowitz RJ | 41720803 | 2024-11-13 | 58440 | |
| 9CX9 | Cryo-EM | 3.3 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Antibody fragment Fab30 Antibody fragment Fab30 |
heavy chain light chain Vasopressin V2 receptor Proto-oncogene tyrosine-protein kinase Src |
- | - | - | Pakharukova N, Thomas BN, Bansia H, Li L, Bassford DK, Abzalimov RR, Kim J, Kahsai AW, Pani B, Xiao K, Ochakovski R, Liu S, Zhang X, Ahn S, des Georges A, Lefkowitz RJ | 41720803 | 2024-11-13 | 58440 | |
| 9DNG | Cryo-EM | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | anti-BRIL Fab Heavy chain anti-BRIL Fab LIGHT chain |
- | - | - | - | Kahsai AW, Pakharukova N, Kwon HY, Shah KS, Del Real CT, Shreiber BN, Liang-Lin JG, Shim PJ, Lee MA, Ngo VA, Schwalb AM, Pham U, Chundi A, Jiang H, Flores-Espinoza E, Liu S, Nibley PC, Bassford DK, Hahn H, Kunzle CA, Thomas BN, Kim J, Zhou Y, Wang J, Zhang X, Smith JS, Rein LAM, Thomsen ARB, Shenoy SK, Rajagopal S, Shi L, Ahn S, Rockman HA, Masoudi A, Lefkowitz RJ | 42343124 | 2025-01-22 | 58440 | |
| 9DNM | Cryo-EM | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | anti-BRIL Fab Heavy chain anti-BRIL Fab Light chain |
- | - | - | - | Kahsai AW, Pakharukova N, Kwon HY, Shah KS, Del Real CT, Shreiber BN, Liang-Lin JG, Shim PJ, Lee MA, Ngo VA, Schwalb AM, Pham U, Chundi A, Jiang H, Flores-Espinoza E, Liu S, Nibley PC, Bassford DK, Hahn H, Kunzle CA, Thomas BN, Kim J, Zhou Y, Wang J, Zhang X, Smith JS, Rein LAM, Thomsen ARB, Shenoy SK, Rajagopal S, Shi L, Ahn S, Rockman HA, Masoudi A, Lefkowitz RJ | 42343124 | 2025-01-22 | 58440 | |
| 9KYU | Cryo-EM | 2.7 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Rat | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C5aR1 phosphopeptide | - | - | - | Mishra S, Yadav MK, Dalal A, Ganguly M, Yadav R, Sawada K, Tiwari D, Roy N, Banerjee N, Fung JN, Marallag J, Cui CS, Li XX, Lee JD, Dsouza CA, Saha S, Sarma P, Rawat G, Zhu H, Khant HA, Clark RJ, Sano FK, Banerjee R, Woodruff TM, Nureki O, Gati C, Shukla AK | 40501890 | 2025-11-26 | 58440 | |
| 2IV8 | X-ray | 2.8 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Human | - | - | - | - | AP-2 complex subunit Beta-1 | - | - | - | Schmid EM, Ford MG, Burtey A, Praefcke GJ, Peak-Chew SY, Mills IG, Benmerah A, McMahon HT | 16903783 | 2007-06-12 | 58438 | |
| 7R0J | Cryo-EM | 4.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Human | - | - | - | ScFv30 | V2R Cter | - | - | - | Bous J, Fouillen A, Orcel H, Trapani S, Cong X, Fontanel S, Saint-Paul J, Lai-Kee-Him J, Urbach S, Sibille N, Sounier R, Granier S, Mouillac B, Bron P | 36054364 | 2022-09-14 | 58438 | |
| 8AS2 | X-ray | 3.2 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Human | - | - | - | Fab30 heavy chain Fab30 light chain |
C-C chemokine receptor type 5 | - | - | - | Isaikina P, Petrovic I, Jakob RP, Sarma P, Ranjan A, Baruah M, Panwalkar V, Maier T, Shukla AK, Grzesiek S | 37244255 | 2023-06-07 | 58438 | |
| 8AS3 | X-ray | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Human | - | - | - | Fab30 heavy chain Fab30 light chain |
C-C chemokine receptor type 5 | - | - | - | Isaikina P, Petrovic I, Jakob RP, Sarma P, Ranjan A, Baruah M, Panwalkar V, Maier T, Shukla AK, Grzesiek S | 37244255 | 2023-06-07 | 58438 | |
| 8AS4 | X-ray | 2.3 | - | - | - | - | - | - | Beta | Beta-arrestin-1 | Human | - | - | - | - | - | - | - | - | Isaikina P, Petrovic I, Jakob RP, Sarma P, Ranjan A, Baruah M, Panwalkar V, Maier T, Shukla AK, Grzesiek S | 37244255 | 2023-06-07 | 58438 | |
| 3P2D | X-ray | 3.0 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | - | - | - | - | - | Zhan X, Gimenez LE, Gurevich VV, Spiller BW | 21215759 | 2011-01-26 | 58474 | |
| 5TV1 | X-ray | 2.4 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | - | - | - | - | - | Chen Q, Perry NA, Vishnivetskiy SA, Berndt S, Gilbert NC, Zhuo Y, Singh PK, Tholen J, Ohi MD, Gurevich EV, Brautigam CA, Klug CS, Gurevich VV, Iverson TM | 29127291 | 2017-11-22 | 58474 | |
| 8GO9 | Cryo-EM | 3.4 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Atypical chemokine receptor 2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58474 | |
| 8GOC | Cryo-EM | 4.2 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Vasopressin V2 receptor | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58474 | |
| 8GOO | Cryo-EM | 4.4 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C5a anaphylatoxin chemotactic receptor 1 | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58474 | |
| 8I0Z | Cryo-EM | 4.3 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C5a anaphylatoxin chemotactic receptor 1 | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58474 | |
| 8I10 | Cryo-EM | 4.0 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Vasopressin V2 receptor | - | - | - | Maharana J, Sarma P, Yadav MK, Saha S, Singh V, Saha S, Chami M, Banerjee R, Shukla AK | 37209686 | 2023-05-17 | 58474 | |
| 8J8R | Cryo-EM | 2.9 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Muscarinic acetylcholine receptor M2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58474 | |
| 8J8V | Cryo-EM | 3.2 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
Atypical chemokine receptor 2 | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58474 | |
| 8TIL | Cryo-EM | 3.8 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab7 heavy chain Fab7 light chain |
Atypical chemokine receptor 3 | - | - | - | Chen Q, Schafer CT, Mukherjee S, Wang K, Gustavsson M, Fuller JR, Tepper K, Lamme TD, Aydin Y, Agrawal P, Terashi G, Yao XQ, Kihara D, Kossiakoff AA, Handel TM, Tesmer JJG | 40399676 | 2025-01-22 | 58474 | |
| 8TIN | Cryo-EM | 4.0 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab7 heavy chain Fab7 light chain |
Atypical chemokine receptor 3 | - | - | - | Chen Q, Schafer CT, Mukherjee S, Wang K, Gustavsson M, Fuller JR, Tepper K, Lamme TD, Aydin Y, Agrawal P, Terashi G, Yao XQ, Kihara D, Kossiakoff AA, Handel TM, Tesmer JJG | 40399676 | 2025-01-22 | 58474 | |
| 8VJ9 | Cryo-EM | 3.3 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab7 heavy chain Fab7 light chain |
Atypical chemokine receptor 3 | - | - | - | Chen Q, Schafer CT, Mukherjee S, Wang K, Gustavsson M, Fuller JR, Tepper K, Lamme TD, Aydin Y, Agrawal P, Terashi G, Yao XQ, Kihara D, Kossiakoff AA, Handel TM, Tesmer JJG | 40399676 | 2025-01-22 | 58474 | |
| 9KY2 | Cryo-EM | 2.8 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Bovine | - | - | - | Fab30 Heavy Chain Fab30 Light Chain |
C5a anaphylatoxin chemotactic receptor 1 | - | - | - | Mishra S, Yadav MK, Dalal A, Ganguly M, Yadav R, Sawada K, Tiwari D, Roy N, Banerjee N, Fung JN, Marallag J, Cui CS, Li XX, Lee JD, Dsouza CA, Saha S, Sarma P, Rawat G, Zhu H, Khant HA, Clark RJ, Sano FK, Banerjee R, Woodruff TM, Nureki O, Gati C, Shukla AK | 40501890 | 2025-11-26 | 58474 | |
| 6K3F | X-ray | 2.3 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Rat | - | - | - | - | Peptide from Atypical chemokine receptor 3 | - | - | - | Min K, Yoon HJ, Park JY, Baidya M, Dwivedi-Agnihotri H, Maharana J, Chaturvedi M, Chung KY, Shukla AK, Lee HH | 32579945 | 2020-06-10 | 58473 | |
| 8J9K | Cryo-EM | 3.5 | - | - | - | - | - | - | Beta | Beta-arrestin-2 | Rat | - | - | - | Fab6 light chain Fab6 heavy chain |
- | - | - | - | Maharana J, Sano FK, Sarma P, Yadav MK, Duan L, Stepniewski TM, Chaturvedi M, Ranjan A, Singh V, Saha S, Mahajan G, Chami M, Shihoya W, Selent J, Chung KY, Banerjee R, Nureki O, Shukla AK | 38175886 | 2023-12-27 | 58473 | |
| 1SUJ | X-ray | 2.4 | - | - | - | - | - | - | Visual | Arrestin-C | Eastern tiger salamander | - | - | - | - | - | - | - | - | Sutton RB, Vishnivetskiy SA, Robert J, Hanson SM, Raman D, Knox BE, Kono M, Navarro J, Gurevich VV | 16289201 | 2005-08-23 | 58502 | |
| 6BK9 | X-ray | 3.0 | - | - | - | - | - | - | Visual | Visual arrestin | Longfin inshore squid | - | - | - | - | - | - | - | - | Bandyopadhyay A, Van Eps N, Eger BT, Rauscher S, Yedidi RS, Moroni T, West GM, Robinson KA, Griffin PR, Mitchell J, Ernst OP | 30120952 | 2018-09-19 | 58521 | |
| 8FUT | X-ray | 2.5 | - | - | - | - | - | - | Visual | S-arrestin | African clawed frog | - | - | - | - | - | - | - | - | Barnes CL, Salom D, Namitz KEW, Smith WC, Knutson BA, Cosgrove MS, Kiser PD, Calvert PD | 39510183 | 2024-07-24 | 58516 | |
| 8FUU | X-ray | 2.9 | - | - | - | - | - | - | Visual | S-arrestin | African clawed frog | - | - | - | - | - | - | - | - | Barnes CL, Salom D, Namitz KEW, Smith WC, Knutson BA, Cosgrove MS, Kiser PD, Calvert PD | 39510183 | 2024-07-24 | 58516 | |
| 1AYR | X-ray | 3.3 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Granzin J, Wilden U, Choe HW, Labahn J, Krafft B, Buldt G | 9495348 | 1998-11-25 | 58515 | |
| 1CF1 | X-ray | 2.8 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Hirsch JA, Schubert C, Gurevich VV, Sigler PB | 10219246 | 1999-04-16 | 58515 | |
| 3UGU | X-ray | 1.9 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Granzin J, Cousin A, Weirauch M, Schlesinger R, Buldt G, Batra-Safferling R | 22306737 | 2012-02-08 | 58515 | |
| 3UGX | X-ray | 2.6 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Granzin J, Cousin A, Weirauch M, Schlesinger R, Buldt G, Batra-Safferling R | 22306737 | 2012-02-08 | 58515 | |
| 4J2Q | X-ray | 3.0 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Kim YJ, Hofmann KP, Ernst OP, Scheerer P, Choe HW, Sommer ME | 23604253 | 2013-05-01 | 58515 | |
| 4ZRG | X-ray | 2.7 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Granzin J, Stadler A, Cousin A, Schlesinger R, Batra-Safferling R | 26510463 | 2015-11-11 | 58515 | |
| 7F1W | X-ray | 3.1 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-27 | 58515 | |
| 7F1X | X-ray | 3.0 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-27 | 58515 | |
| 7JSM | X-ray | 2.5 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7JTB | X-ray | 2.6 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7JXA | X-ray | 2.4 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7MOR | X-ray | 2.8 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7MP0 | X-ray | 2.6 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7MP1 | X-ray | 2.7 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 7MP2 | X-ray | 3.0 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Sander CL, Luu J, Kim K, Furkert D, Jang K, Reichenwallner J, Kang M, Lee HJ, Eger BT, Choe HW, Fiedler D, Ernst OP, Kim YJ, Palczewski K, Kiser PD | 34678158 | 2021-10-13 | 58515 | |
| 9C6E | X-ray | 1.4 | - | - | - | - | - | - | Visual | S-arrestin | Bovine | - | - | - | - | - | - | - | - | Salom D, Kiser PD, Palczewski K | 39704710 | 2024-11-06 | 58515 | |
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